China (Mainland)
K252a CAS NO.99533-80-9
- Min.Order: 0 Metric Ton
- Payment Terms: T/T
- Product Details
Keywords
- 99533-80-9
- K252a
- K252a, in stock
Quick Details
- ProName: K252a
- CasNo: 99533-80-9
- Molecular Formula: C27H21N3O5
- Appearance: Off-white to light yellow (Solid)
- Application: Protein and CAM kinases inhibitor;Anti...
- DeliveryTime: In stock
- PackAge: As per request
- Port: Shanghai
- ProductionCapacity: Metric Ton/Day
- Purity: 90%+
- Storage: Store in a tight container at -20℃.
- Transportation: by air or by sea
- LimitNum: 0 Metric Ton
Superiority
Product in stock
Short lead time
Cost competitiveness
Details
K-252a, a staurosporine analog isolated from Nocardiopsis sp. soil fungi, inhibits protein kinase, with IC50 values of 470 nM, 140 nM, 270 nM, and 1.7 nM for PKC, PKA, Ca2+/calmodulin-dependent kinase type II, and phosphorylase kinase, respectively. K-252a is a potent inhibitor (IC50 of 3 nM) of the tyrosine protein kinase (TRK) activity of the NGF receptor gp140trk, the product of the trk protooncogene.